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GIUSEPPE DAIDONE

Pubblicazioni

Data Titolo Tipologia Scheda
2019 Novel 4-(3-phenylpropionamido), 4-(2-phenoxyacetamido) and 4-(cinnamamido) substituted benzamides bearing the pyrazole or indazole nucleus: synthesis, biological evaluation and mechanism of action Articolo in rivista Vai
2018 Sintesi e valutazione biologica di nuovi nitroderivati analoghi della pirrolomicina D attivi su Pseudomonas aeruginosa Proceedings (TIPOLOGIA NON ATTIVA) Vai
2018 Sintesi di un isostero del 3,5-dimetil-6-fenil-8-(trifluorometil)-5,6-diidropirazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one (CF3-TZP) con potenziale attività biologica Proceedings (TIPOLOGIA NON ATTIVA) Vai
2018 Progettazione e sintesi di nuovi derivati 4-chinazolinonici potenziali inibitori della diidrofolato reduttasi Proceedings (TIPOLOGIA NON ATTIVA) Vai
2018 The role of (E)-6-chloro-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-styrylquinazolin-4(3H)-one in the modulation of cannabinoidergic system. A pilot study Articolo in rivista Vai
2018 Pirrolomicine che inibiscono la Sortasi A nelle infezioni sostenute da batteri Gram-positivi Proceedings (TIPOLOGIA NON ATTIVA) Vai
2017 Recent discoveries of anticancer flavonoids Articolo in rivista Vai
2017 Anthranilamide-based 2-phenylcyclopropane-1-carboxamides, 1,1'-biphenyl-4-carboxamides and 1,1'-biphenyl-2-carboxamides: Synthesis biological evaluation and mechanism of action Articolo in rivista Vai
2017 The Reactivity of 4’-Substituted Spiro[Isoindole-1,3’-pyrazoles] Derivatives: Substitution/Elimination Reactions and Access to Biaryl Derivatives Articolo in rivista Vai
2017 Derivati policiclici con struttura complessa dotati di attività antiproliferativa Proceedings (TIPOLOGIA NON ATTIVA) Vai
2016 A new class of phenylhydrazinylidene derivatives as inhibitors of Staphylococcus aureus biofilm formation Articolo in rivista Vai
2016 Discovery of a new class of sortase a transpeptidase inhibitors to tackle gram-positive pathogens: 2-(2-phenylhydrazinylidene)alkanoic acids and related derivatives Articolo in rivista Vai
2016 Isoxazolo[3,4-d]pyridazin-7(6H)-one derivatives endowed with anti-proliferative Activity. Proceedings (TIPOLOGIA NON ATTIVA) Vai
2016 Synthesis and antiproliferative activities of two new analogs of tetrazepinones Proceedings (TIPOLOGIA NON ATTIVA) Vai
2016 Synthesized benzamido derivatives exert antiproliferative effects by DNA damage and ROS generation. Proceedings (TIPOLOGIA NON ATTIVA) Vai
2016 Synthesis and antiproliferative activity of a natural like glycoconjugate polycyclic compound Articolo in rivista Vai
2016 Synthesis and biofilm formation reduction of pyrazole-4-carboxamide derivatives in some Staphylococcus aureus strains Articolo in rivista Vai
2015 Recent advanced in bioactive systems containing pyrazole fused with a five membered heterocycle Articolo in rivista Vai
2015 Sortase A Inhibitors: Recent Advances and Future Perspectives Articolo in rivista Vai
2015 New Anti-Adhesion Agents In The Development of Antivirulence Drugs Proceedings (TIPOLOGIA NON ATTIVA) Vai
2015 Pharmaceutical Potential of Synthetic and Natural Pyrrolomycins Articolo in rivista Vai
2015 Synthesis, antiproliferative activity and possible mechanism of action of novel 2-acetamidobenzamides bearing the 2-phenoxy functionality Articolo in rivista Vai
2015 Synthesis and antiproliferative activity of 3-(2-cloroethyl)-5-methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-(3H)-one Articolo in rivista Vai
2015 Discovery of a New Class of Sortase A Transpeptidase Inhibitors to Tackle Gram-positive Pathogens: 2-Phenylhydrazonoalkanoic Acid Derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2014 Synthesis and antiproliferative activity of a natural like glucosyl polycyclic compound Proceedings (TIPOLOGIA NON ATTIVA) Vai
2014 NUOVI DERIVATI 2-ACETAMMIDOBENZAMMIDICI: ATTIVITÀ ANTIPROLIFERATIVA E POSSIBILE MECCANISMO DI AZIONE Proceedings (TIPOLOGIA NON ATTIVA) Vai
2014 RADICAL CYCLIZATION AND 1,5-HYDROGEN TRANSFER IN SELECTED AROMATIC DIAZONIUM SALTS Articolo in rivista Vai
2014 Synthesis and antiproliferative activity of new derivatives containing the polycyclic system 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3’,4’:2,3]azepino[4,5-f]azocine Articolo in rivista Vai
2014 ATTIVITÀ ANTIPROLIFERATIVA DI UN DERIVATO POLICICLICO CON STRUTTURA COMPLESSA Proceedings (TIPOLOGIA NON ATTIVA) Vai
2014 Unexpected synthesis by a non-classical Pschorr reaction of 3,5-dimethyl-1-phenyl-1,5-dihydro-4H-pyrazolo[4,3-c]quinolin-4-one, with binding affinity for the central benzodiazepine receptor Articolo in rivista Vai
2014 Synthesis and antirpoliferative activity of isoxazolo[3,4-d]pyridazin-7(6H)-one derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2013 2-Cinnamamido, 2-(3-phenylpropiolamido), and 2-(3-phenylpropanamido)benzamides: synthesis, antiproliferative activity, and mechanism of action Articolo in rivista Vai
2013 Non-Classical Transformation of Benzendiazonium Hydrogen Sulfates. Access to 1,3-Dimethylisochromeno[4,3-c]pyrazol-5(1H)-one, a Potential Benzodiazepine Receptor Ligand Articolo in rivista Vai
2013 2-cinnamamido, 2-(3-phenylpropiolamido) and 2-(3-phenylpropanamido)benzamides: synthesis, antiproliferative activity and mechanism of action Proceedings (TIPOLOGIA NON ATTIVA) Vai
2013 Novel Sortase A (SrtA) inhibitors interfere with the formation of staphylococcal biofilms Proceedings (TIPOLOGIA NON ATTIVA) Vai
2012 Synthesis and antioproliferative activity of new derivatives containing the policyclic sistem 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3'.4':2,3]azepino[4,5-f]azocine Proceedings (TIPOLOGIA NON ATTIVA) Vai
2012 Synthesis, benzodiazepine receptor binding and molecular modelling of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives Articolo in rivista Vai
2012 Synthesis and anti-staphylococcal activity of new 4-diazopyrazole derivatives Articolo in rivista Vai
2011 Synthesis and antiproliferative activity of indazole derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2011 Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[2E]-3-phenylprop-2-enoylamino}benzamides Articolo in rivista Vai
2011 Synthesis, antiproliferative activity, and mechanism of action of new benzamido derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2011 Synthesis of substituted 3-amino-N-phenyl-1H-indazole-1-carboxamides endowed with antiproliferative activity Articolo in rivista Vai
2010 NEW 4-DIAZOPYRAZOLE DERIVATIVES AS POTENTIAL ANTIBIOFILM AGENTS Proceedings (TIPOLOGIA NON ATTIVA) Vai
2010 Reazioni consecutive di Pschorr e Sandmeyer non classiche in serie isossazolica. Accesso a composti di interesse farmaceutico Proceedings (TIPOLOGIA NON ATTIVA) Vai
2010 Synthesis and biological evaluation of new indazole derivatives Articolo in rivista Vai
2010 Reazioni consecutive di Pschorr e Sandmeyer non classiche in serie pirazolo-tiofenica. Accesso a composti di interesse farmaceutico Proceedings (TIPOLOGIA NON ATTIVA) Vai
2010 SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF 3-AMINO-N-PHENYL-1H-INDAZOLE-1-CARBOXAMIDES Proceedings (TIPOLOGIA NON ATTIVA) Vai
2009 N-(INDAZOLYL)BENZAMIDO DERIVATIVES AS CDK1 INHIBITORS: DESIGN, SYNTHESIS, BIOLOGICAL ACTIVITY, AND MOLECULAR DOCKING STUDIES Articolo in rivista Vai
2009 Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamides Articolo in rivista Vai
2009 5-Amino-1-phenyl-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid Articolo in rivista Vai
2008 4-Diazopyrazole Derivatives as Potential New Antibiofilm Agents Articolo in rivista Vai
2008 1,4-Dimethyl-3-phenyl-3H-pyrazolo[3,4-c]isoquinolin-5(4H)-one Articolo in rivista Vai
2008 Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one Articolo in rivista Vai
2008 Comparative studies of the Pschorr reaction in the pyrazole series. Access to the new dibenzo(e,g)pyrazolo(1,5-a)(1,3)diazocine system of pharmaceutical interest Articolo in rivista Vai
2008 SYNTHESIS AND BIOLOGICAL EVALUATION OF 2-PHENYL-3-[INDAZOL-3-YL]-4(3H)-QUINAZOLINONES Proceedings (TIPOLOGIA NON ATTIVA) Vai
2007 Synthesis and biological activity of new anti-inflammatory compounds containing the 1,4-benzodioxine and/or pyrrole system Articolo in rivista Vai
2007 Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-trifluoromethyl-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-one Proceedings (TIPOLOGIA NON ATTIVA) Vai
2007 Synthesis and biological evaluation of new 2-{[(2E)-3-phenylprop-2-enoyl]amino}benzamides Proceedings (TIPOLOGIA NON ATTIVA) Vai
2007 Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamide derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2007 Antileukemic activity of some new 3-amino-N-phenyl-(1H)-indazole-1-carboxamide derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2007 Synthesis and anticancer activity of 3-amino-N-phenyl-1H-indazole-1-carboxamide and 1-(1H)indazol-3-yl-3-phenylureido derivatives Proceedings (TIPOLOGIA NON ATTIVA) Vai
2006 Synthesis of New Pyrazole Derivatives as Potential CDK1 Inhibitors Proceedings (TIPOLOGIA NON ATTIVA) Vai
2006 Synthesis and Antiproliferative Activity of a New Pyrazolo[3,4-f]1,2,3,5-tetrazepin-4(3H)-one Derivative Proceedings (TIPOLOGIA NON ATTIVA) Vai
2006 Synthesis of alkyl-5,8-dimethyl-6-phenyl-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-ones of pharmaceutical interest Articolo in rivista Vai
2005 Nonclassical Pschorr and Sandmeyer Reactions in Pyrazole Series Articolo in rivista Vai
2005 BENZOTRIAZINONE AND QUINAZOLINONE DERIVATIVES AS COX-INHIBITORS: COMPUTATIONAL STUDIES Proceedings (TIPOLOGIA NON ATTIVA) Vai
2005 Comparative Structural Studies of 4-Diazopyrazole Derivatives by X-Ray Diffraction and Theoretical Investigation Articolo in rivista Vai
2005 Unclassical Pschorr and Sandmeyer reactions in pyrazole series Proceedings (TIPOLOGIA NON ATTIVA) Vai
2004 Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones. Articolo in rivista Vai
2004 SYNTHESIS AND IN VITRO ANTILEUKEMIC ACTIVITY OF NEW 4-TRIAZENOPYRAZOLE DERIVATIVES Articolo in rivista Vai
2004 SINTESI ED ATTIVITÀ ANTINEOPLASTICA DI NUOVI COMPOSTI ETEROCICLICI Tesi di dottorato pre 2013 Vai
2004 SYNTHESIS AND ANTILEUKEMIC ACTIVITY OF NEW 3-(1-PHENYL-3-METHYLPYRAZOL-5-YL)-2-STYRYLQUINAZOLIN-4(3H)-ONES Articolo in rivista Vai
2004 SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF TRIAZENOINDAZOLES AND TRIAZENOPYRAZOLES: A COMPARATIVE STUDY Articolo in rivista Vai
2004 SYNTHESIS, CYTOTOXICITY, AND INHIBITORY EFFECTS ON TUBULIN POLYMERIZATION OF A NEW 3-HETEROCYCLO SUBSTITUTED 2-STYRYLQUINAZOLINONES Articolo in rivista Vai
2002 Synthesis and antifungal activity of new N-(1-phenil-4-carbetoxypyrazol-5-yl)-N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides Articolo in rivista Vai
1999 Synthesis and antifungal activity of new N-isoxazolyl-2-iodobenzamides Articolo in rivista Vai